SCHEMBL9857802

SCHEMBL9857802

Cc1cc(-c2cc(-c3ccccc3)cc(C)c2C=O)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.44
PTGS1 P23219 2/20 0.43
DAPK3 O43293 1/20 0.37
NTRK1 P04629 1/20 0.37
PIM1 P11309 1/20 0.37
FLT3 P36888 1/20 0.37
GSK3B P49841 1/20 0.37
ROCK1 Q13464 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
BRD4 O60885 1/20 0.36
HPRT1 P00492 1/20 0.36
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
SRC P12931 1/20 0.35
KAT6A Q92794 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857896 0.87 PTGS2 (0.39) PTGS2PTGS1
SCHEMBL9857094 0.87 PTGS2 (0.41) PTGS2PTGS1BRD4HPRT1TNKS2
SCHEMBL5171500 0.83 PTGS2 (0.48) PTGS2PTGS1DAPK3NTRK1PIM1
SCHEMBL10741025 0.82 PTGS2 (0.47) PTGS2PTGS1DAPK3NTRK1PIM1
SCHEMBL15676174 0.79 BRD4 (0.42) PTGS2BRD4TNKS2
SCHEMBL5762155 0.77 ACHE (0.48) PTGS2PTGS1DAPK3NTRK1PIM1
SCHEMBL9857622 0.77 AKR1C2 (0.42) PTGS2PTGS1SRCKAT6A
SCHEMBL28930334 0.74 PTGS2 (0.40) PTGS2PTGS1DAPK3NTRK1PIM1
SCHEMBL9857687 0.73 PTGS2 (0.41) PTGS2PTGS1HPRT1SRC
SCHEMBL10742738 0.73 MEN1 (0.46) PTGS2PTGS1TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072023-A Reacting lactone with ester anion to form cyclohexenone ester; oxidizing or dehydrogenating the intermediate E. R. SQUIBB & SONS, INC. (US) 1991-12-10 US disclosed
EP-0442495-A1 Process for preparing highly substituted phenyls E.R. SQUIBB & SONS, INC. (US) 1991-08-21 EP disclosed