SCHEMBL9857778

SCHEMBL9857778

O=C(NC=C(c1ccccc1)c1ccccc1)c1sc2ccc(F)cc2c1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
RAB9A P51151 3/20 0.39
GAA P10253 2/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
HSP90AA1 P07900 1/20 0.39
TNNI3 P19429 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
TNNT2 P45379 1/20 0.39
TNNC1 P63316 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
LRRK2 Q5S007 1/20 0.39
PMM2 O15305 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10624313 0.84 LRRK2 (0.39) MEN1KMT2ARAB9AGAANPC1
SCHEMBL9858136 0.84 RAB9A (0.40) MEN1KMT2ARAB9AGAANPC1
SCHEMBL9857661 0.82 KDM4E (0.40) RAB9AGAANPC1MAPTKDM4E
SCHEMBL9857258 0.81 RAB9A (0.38) MEN1KMT2ARAB9AGAANPC1
SCHEMBL9857207 0.78 MAOB (0.45) MEN1KMT2ARAB9AGAANPC1
SCHEMBL9857203 0.78 MAOB (0.45) MEN1KMT2ARAB9AGAANPC1
SCHEMBL10681141 0.76 RAB9A (0.38) MEN1KMT2ARAB9ANPC1KDM4E
SCHEMBL6008817 0.76 RAB9A (0.38) MEN1KMT2ARAB9ANPC1KDM4E
SCHEMBL9857805 0.76 KDM4E (0.40) MEN1KMT2ARAB9ANPC1MAPT
SCHEMBL9857650 0.76 TSHR (0.39) MEN1KMT2ARAB9AGAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068248-A Analgesics, antipyretics and antiinflammatory agents MERCK & CO., INC. (US) 1991-11-26 US disclosed
EP-0160408-B1 BENZOTHIOPHENES, THEIR PRODUCTION AND USE, AND COMPOSITIONS CONTAINING THEM MERCK & CO. INC. (US) 1989-08-23 EP disclosed
US-4760086-A N-alkenyl-3-hydroxybenzo[b]thiophene-2-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-07-26 US disclosed
EP-0160408-A1 Benzothiophenes, their production and use, and compositions containing them MERCK & CO. INC. (US) 1985-11-06 EP disclosed