SCHEMBL9858136

SCHEMBL9858136

CSc1ccc2sc(C(=O)NC=C(c3ccccc3)c3ccccc3)c(O)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.40
KMT2A Q03164 7/20 0.40
NPC1 O15118 7/20 0.40
MEN1 O00255 6/20 0.40
GAA P10253 3/20 0.40
MAOB P27338 4/20 0.36
MAOA P21397 1/20 0.36
SMN1; SMN2 Q16637 7/20 0.36
MAPT P10636 7/20 0.36
ALPG P10696 1/20 0.36
KDM4E B2RXH2 4/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
LMNA P02545 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
HSP90AA1 P07900 1/20 0.35
TNNI3 P19429 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857778 0.84 MEN1 (0.39) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL9857258 0.81 RAB9A (0.38) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL10624497 0.80 KMT2A (0.35) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL10624501 0.80 KMT2A (0.35) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL9857661 0.78 KDM4E (0.40) RAB9ANPC1GAAMAPTKDM4E
SCHEMBL10629092 0.77 SMN1; SMN2 (0.33) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL10481451 0.77 PTGS2 (0.58) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL9857207 0.77 MAOB (0.45) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL9857203 0.77 MAOB (0.45) RAB9AKMT2ANPC1MEN1GAA
SCHEMBL10626989 0.74 CCR2 (0.38) RAB9AKMT2ANPC1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068248-A Analgesics, antipyretics and antiinflammatory agents MERCK & CO., INC. (US) 1991-11-26 US disclosed
US-4760086-A N-alkenyl-3-hydroxybenzo[b]thiophene-2-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-07-26 US disclosed
EP-0160408-A1 Benzothiophenes, their production and use, and compositions containing them MERCK & CO. INC. (US) 1985-11-06 EP disclosed