SCHEMBL9857795

SCHEMBL9857795

O=C(CCl)NCC(O)(c1ccccc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
HTT P42858 6/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
MITF O75030 1/20 0.42
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
CNR1 P21554 2/20 0.41
CNR2 P34972 2/20 0.41
OGT O15294 1/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
MAPK1 P28482 2/20 0.39
XBP1 P17861 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
RNF4 P78317 1/20 0.39
TRPA1 O75762 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5967138 0.82 CYP1A2 (0.46) MEN1KMT2ACNR1CNR2MAPK1
SCHEMBL2065478 0.81 MEN1 (0.50) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL9354938 0.81 CNR1 (0.42) ALDH1A1HTTSMN1; SMN2RAB9ANPC1
SCHEMBL3901654 0.78 LMNA (0.48) HTTSMN1; SMN2MEN1KMT2ACNR1
SCHEMBL31322256 0.75 CYP2C19 (0.42) ALDH1A1HTTSMN1; SMN2RAB9ANPC1
SCHEMBL6599652 0.74 SMN1; SMN2 (0.51) ALDH1A1HTTSMN1; SMN2RAB9ANPC1
SCHEMBL11409037 0.72 ALDH1A1 (0.56) ALDH1A1MEN1KMT2ALMNAKDM4E
SCHEMBL11409035 0.72 ALDH1A1 (0.56) ALDH1A1MEN1KMT2ALMNAKDM4E
SCHEMBL1389497 0.71 KIF11 (0.47) ALDH1A1SMN1; SMN2RAB9ANPC1
SCHEMBL2067960 0.71 IDO1 (0.46) RAB9ANPC1MEN1KMT2AHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068248-A Analgesics, antipyretics and antiinflammatory agents MERCK & CO., INC. (US) 1991-11-26 US disclosed
EP-0160408-B1 BENZOTHIOPHENES, THEIR PRODUCTION AND USE, AND COMPOSITIONS CONTAINING THEM MERCK & CO. INC. (US) 1989-08-23 EP disclosed
US-4760086-A N-alkenyl-3-hydroxybenzo[b]thiophene-2-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-07-26 US disclosed
EP-0160408-A1 Benzothiophenes, their production and use, and compositions containing them MERCK & CO. INC. (US) 1985-11-06 EP disclosed