SCHEMBL9861355

SCHEMBL9861355

Cc1cc(C(F)(F)F)cc(C(C)(C)C)c1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.50
RAPGEF4 Q8WZA2 3/20 0.39
CACNA1H O95180 2/20 0.36
CACNA1G O43497 1/20 0.36
CACNA1C Q13936 1/20 0.36
ALDH1A1 P00352 3/20 0.36
TSHR P16473 2/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CA2 P00918 1/20 0.35
TYR P14679 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KIF11 P52732 1/20 0.35
IKBKB O14920 1/20 0.35
PDE2A O00408 1/20 0.35
AR P10275 1/20 0.33
MAPK1 P28482 1/20 0.33
NR2E1 Q9Y466 1/20 0.33
PTPN5 P54829 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861535 0.89 POLB (0.39) POLBCACNA1HCACNA1GCACNA1CALDH1A1
SCHEMBL21615516 0.87 POLB (0.43) POLBRAPGEF4CACNA1HCACNA1GCACNA1C
SCHEMBL10342450 0.85 POLB (0.70) POLBALDH1A1TSHRTP53CYP3A4
SCHEMBL9861925 0.83 POLB (0.61) POLBALDH1A1TSHRTP53CYP3A4
SCHEMBL532346 0.82 POLB (0.56) POLBRAPGEF4ALDH1A1TSHRTP53
Hydrochloric Acid SCHEMBL19857169 0.80 POLB (0.61) POLBRAPGEF4ALDH1A1TSHRTP53
SCHEMBL9861913 0.80 POLB (0.42) POLBALDH1A1TSHRTP53CYP3A4
SCHEMBL25767375 0.78 RAPGEF4 (0.37) POLBRAPGEF4CACNA1HCACNA1GCACNA1C
SCHEMBL16022232 0.78 ALDH1A1 (0.52) POLBRAPGEF4ALDH1A1TSHRTP53
SCHEMBL8943131 0.78 POLB (0.65) POLBALDH1A1TSHRTP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed