SCHEMBL9861457

SCHEMBL9861457

CCOc1cccc2c1C(O[Si](CC)(CC)CC)(C(F)(F)C(F)(F)F)C(=O)c1ccccc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.39
MAPT P10636 2/20 0.38
ALPL P05186 1/20 0.36
PTPRC P08575 1/20 0.36
ALDH1A1 P00352 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
HPGD P15428 1/20 0.34
KCNK3 O14649 1/20 0.34
KCNK9 Q9NPC2 1/20 0.34
GRM5 P41594 1/20 0.34
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
GUSB P08236 1/20 0.33
TRPA1 O75762 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
APAF1 O14727 1/20 0.32
USP2 O75604 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861411 0.81 S100A4 (0.36) PDK2
SCHEMBL9861482 0.77 PDK2 (0.51) PDK2MAPTALPLPTPRCALDH1A1
SCHEMBL9861632 0.73 S100A4 (0.38) PDK2
SCHEMBL9861961 0.73 KCNQ2 (0.40) PDK2
SCHEMBL9861564 0.67 ADORA2A (0.36) PDK2MAPTPTPRCALDH1A1L3MBTL1
SCHEMBL9861333 0.65 KCNQ2 (0.42) PDK2
SCHEMBL9861915 0.64 MEN1 (0.36) PDK2MAPTALDH1A1L3MBTL1HPGD
SCHEMBL18723280 0.60 L3MBTL1 (0.50) PDK2MAPTALDH1A1L3MBTL1HPGD
SCHEMBL14940040 0.59 CYP2D6 (0.45) PDK2MAPTPTPRCALDH1A1L3MBTL1
SCHEMBL198911 0.59 ALDH1A1 (0.60) MAPTPTPRCALDH1A1L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4844892-A MOSQUITOES NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4803289-A MOSQUITOES NATIONAL RESEARCH DEVELOPMENT CORP. (GB) 1989-02-07 US disclosed
EP-0078641-B1 IMPROVEMENTS IN OR RELATING TO PHEROMONES NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1986-02-26 EP disclosed
EP-0078641-A1 Improvements in or relating to pheromones NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1983-05-11 EP disclosed
WO-1983001621-A1 IMPROVEMENTS IN OR RELATING TO PHEROMONES LAURENCE, BRIAN, ROBIN 1983-05-11 WO disclosed