SCHEMBL9861499

SCHEMBL9861499

CCc1cc(C(F)(F)C(F)(F)C(F)(F)F)c2ccccc2c1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 3/20 0.46
MAPT P10636 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPK1 P28482 2/20 0.46
HTT P42858 2/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PGR P06401 7/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
GLA P06280 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
ATM Q13315 1/20 0.36
EP300 Q09472 1/20 0.34
NPY5R Q15761 1/20 0.33
ELANE P08246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861455 0.84 KDM4E (0.44) KDM4EMEN1MAPTKMT2AMAPK1
SCHEMBL9862072 0.83 GABRA1 (0.40) KDM4EMEN1MAPTKMT2AMAPK1
SCHEMBL5958646 0.72 HTT (0.40) MAPTHTTPGRALDH1A1POLB
SCHEMBL9778555 0.71 PKM (0.42) KDM4EMEN1MAPTKMT2AMAPK1
SCHEMBL9861512 0.69 KDM4E (0.53) KDM4EMEN1MAPTKMT2AMAPK1
SCHEMBL28883537 0.68 CYP1A2 (0.39) KDM4EMEN1MAPTKMT2AMAPK1
SCHEMBL9861302 0.68 KDM4E (0.60) KDM4EMEN1MAPTKMT2AMAPK1
SCHEMBL9861301 0.68 GABRA1 (0.44) PGRGABRA1GABRB2AR
SCHEMBL3819583 0.68 HMGB1 (0.47) KDM4EMEN1KMT2ALMNAALDH1A1
SCHEMBL5958697 0.67 HTT (0.39) MAPTHTTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed