SCHEMBL9861508

SCHEMBL9861508

CCCCCCC(C)c1cc(C(F)(F)F)c2ccccc2c1N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.36
KDM4E B2RXH2 3/20 0.35
MAPT P10636 2/20 0.35
KMT2A Q03164 2/20 0.35
BACE1 P56817 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
AR P10275 1/20 0.34
TLR8 Q9NR97 1/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
CSNK1E P49674 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861924 0.87 KDM4E (0.36) KCNH2KDM4EMAPTKMT2AMEN1
SCHEMBL9861556 0.85 KCNH2 (0.38) KCNH2KDM4EKMT2ASPHK2SPHK1
SCHEMBL9861970 0.79 P2RX7 (0.38) KCNH2MAPTMAPK1SMN1; SMN2TLR8
SCHEMBL19406660 0.78 CYP1A2 (0.39) KCNH2MAPTMAPK1SMN1; SMN2TLR8
SCHEMBL9861337 0.77 KDM4E (0.44) KDM4EMAPTKMT2ABACE1MEN1
SCHEMBL16442414 0.76 CYP1A2 (0.39) KCNH2MAPTMAPK1SMN1; SMN2TLR8
SCHEMBL9232277 0.76 CYP1A2 (0.39) KCNH2MAPTMAPK1SMN1; SMN2TLR8
SCHEMBL30857800 0.74 AR (0.33) KCNH2ARTLR8ADRB2
SCHEMBL9861423 0.73 GPR84 (0.34) KCNH2KDM4EKMT2APSEN1PSEN2
SCHEMBL30220388 0.72 TLR8 (0.41) KDM4EKMT2AMEN1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed