SCHEMBL9863446

SCHEMBL9863446

CC([N])Cc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.58
SIGMAR1 Q99720 5/20 0.58
SLC6A2 P23975 3/20 0.58
SLC6A4 P31645 2/20 0.58
SLC6A3 Q01959 2/20 0.58
MAOA P21397 1/20 0.58
CYP2A6 P11509 1/20 0.58
ADORA2A P29274 1/20 0.58
ADORA1 P30542 1/20 0.58
SLC18A2 Q05940 1/20 0.54
CYP2D6 P10635 1/20 0.54
TRPA1 O75762 2/20 0.52
EPHX1 P07099 1/20 0.50
TDP1 Q9NUW8 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
HTR2A P28223 1/20 0.48
ADRA1A P35348 1/20 0.48
OPRK1 P41145 1/20 0.48
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30934 0.78 TRPA1 (0.77) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL4785594 0.78 SIGMAR1 (0.64) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
Isobutylbenzene SCHEMBL2571645 0.78 SIGMAR1 (0.64) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
Isobutylbenzene SCHEMBL57393 0.78 SIGMAR1 (0.64) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
Isobutylbenzene SCHEMBL7493657 0.78 SIGMAR1 (0.64) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
Isobutylbenzene SCHEMBL11736259 0.77 TAAR1 (0.56) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL1140503 0.76 TRPA1 (0.74) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
Isobutylbenzene SCHEMBL11468970 0.76 TAAR1 (0.61) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
Water SCHEMBL3896311 0.76 TRPA1 (0.74) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3
Isobutylbenzene SCHEMBL6891614 0.76 SIGMAR1 (0.61) TAAR1SIGMAR1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5025005-A Preventive or therapeutic agents for circulatory diseases, allergic disorders; antineoplastic agent; inhibitor for platelet activating factor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-06-18 US disclosed
US-4737518-A ANTIALLERGENS, ANTINEOPLASTICS, ANTICOAGULANTS, CIRCULATORY DISEASES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-04-12 US disclosed
EP-0157609-A2 Lipid derivatives their production and use Takeda Chemical Industries, Ltd. (JP) 1985-10-09 EP disclosed