SCHEMBL9864486

SCHEMBL9864486

N#CCC(=O)c1ccc(CCc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.51
GSK3B P49841 1/20 0.51
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
DAO P14920 1/20 0.47
MMP1 P03956 1/20 0.45
SRD5A2 P31213 1/20 0.45
HDAC1 Q13547 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
TAAR1 Q96RJ0 1/20 0.43
PDPK1 O15530 1/20 0.43
HSD11B1 P28845 1/20 0.42
VNN1 O95497 1/20 0.41
MMP2 P08253 1/20 0.41
MMP8 P22894 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL133449 0.92 PTPN1 (0.59) PTPN1GSK3BCES2CES1MMP1
SCHEMBL30737605 0.84 LSS (0.60) HDAC1
SCHEMBL5644564 0.79 FFAR1 (0.48) CES2CES1DAOSRD5A2HDAC1
SCHEMBL395103 0.77 GSK3B (0.48) PTPN1GSK3BCES1
SCHEMBL5793959 0.77 L3MBTL1 (0.57)
SCHEMBL28150824 0.76 SRD5A2 (0.72) PTPN1GSK3BCES2CES1SRD5A2
SCHEMBL28166342 0.76 FFAR1 (0.52) SRD5A2
SCHEMBL4306951 0.75 CES2 (0.59) PTPN1GSK3BCES2CES1HDAC8
SCHEMBL393300 0.75 RAB9A (0.56) SRD5A2HDAC1
SCHEMBL4847457 0.74 PTPN1 (0.63) PTPN1GSK3BCES2CES1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0407955-A1 New hetrazepines acting as PAF antagonists, process for their production and their use as drugs BOEHRINGER INGELHEIM KG (DE) 1991-01-16 EP disclosed