SCHEMBL9864882

SCHEMBL9864882

CSC(SC)=C(C#N)c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPK1 P28482 2/20 0.39
TSHR P16473 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CYP3A4 P08684 1/20 0.39
ATM Q13315 1/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 3/20 0.39
RAB9A P51151 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 1/20 0.39
XBP1 P17861 1/20 0.39
CES2 O00748 2/20 0.35
CES1 P23141 2/20 0.35
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865224 0.80 HDAC3 (0.41) MEN1KMT2AMAPK1TSHRALDH1A1
SCHEMBL11566324 0.78 THRB (0.40) MEN1KMT2AMAPK1TSHRL3MBTL1
SCHEMBL9864429 0.78 MEN1 (0.35) MEN1KMT2AL3MBTL1ALDH1A1MAPT
SCHEMBL9864434 0.78 MEN1 (0.35) MEN1KMT2AL3MBTL1ALDH1A1MAPT
SCHEMBL31552934 0.78 DGAT1 (0.48) MEN1KMT2AMAPK1L3MBTL1ALDH1A1
SCHEMBL8022899 0.76 TSHR (0.41) MEN1KMT2AMAPK1TSHRL3MBTL1
SCHEMBL2443924 0.75 NPSR1 (0.71) MEN1KMT2AMAPK1TSHRL3MBTL1
SCHEMBL8032317 0.70 CES2 (0.48) MEN1KMT2ATSHRL3MBTL1CYP3A4
SCHEMBL8032319 0.70 CES2 (0.48) MEN1KMT2ATSHRL3MBTL1CYP3A4
SCHEMBL8022876 0.69 CES2 (0.48) MEN1KMT2ATSHRL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994485-A Seed and soil fungi, bacteria DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1991-02-19 US disclosed
EP-0234622-B1 NEW THIO COMPOUNDS HAVING FUNGICIDAL ACTIVITY DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-06-27 EP disclosed
EP-0234622-A1 New thio compounds having fungicidal activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1987-09-02 EP disclosed