SCHEMBL9866288

SCHEMBL9866288

CC(CSCc1ccccc1)NC(=N)NCCCc1c[nH]cn1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 6/20 0.37
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2D6 P10635 1/20 0.35
KMT2A Q03164 1/20 0.35
ACE P12821 1/20 0.34
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SIGMAR1 Q99720 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867255 0.89 ALDH1A1 (0.37) CYP2C19KMT2ACYP1A2POLBNPSR1
SCHEMBL9866816 0.83 SLC47A1 (0.36) CYP2C19CYP2D6KMT2ACYP1A2SMN1; SMN2
SCHEMBL9866194 0.83 SLC47A1 (0.36) CYP2C19CYP2D6KMT2ACYP1A2SMN1; SMN2
SCHEMBL10872563 0.83
SCHEMBL9866169 0.83 SLC47A1 (0.36) CYP2C19CYP2D6KMT2ACYP1A2SMN1; SMN2
Hydrochloric Acid SCHEMBL9865304 0.82 L3MBTL1 (0.37) CYP2C19CYP2D6KMT2ACYP1A2SMN1; SMN2
Hydrochloric Acid SCHEMBL9866175 0.82 L3MBTL1 (0.37) CYP2C19CYP2D6KMT2ACYP1A2SMN1; SMN2
Hydrochloric Acid SCHEMBL10874476 0.82 L3MBTL1 (0.37) CYP2C19CYP2D6KMT2ACYP1A2SMN1; SMN2
SCHEMBL9866870 0.81 MTNR1A (0.44) CYP2C19CYP2D6KMT2ACYP1A2ALDH1A1
SCHEMBL9866299 0.81 HRH4 (0.37) EPHX2CYP2C9CYP2C19CYP2D6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021431-A H-1 antagonist, h-2 agonist for treating hypertension, cardiac disease or arterial occlusion HEUMANN PHARMA GMBH & CO. (DE) 1991-06-04 US disclosed
EP-0199845-B1 IMIDAZOLYLALKYLGUANIDIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM HEUMANN PHARMA GMBH & CO (DE) 1990-08-01 EP disclosed
EP-0199845-A1 Imidazolylalkylguanidin derivatives, process for their preparation and pharmaceutical compositions containing them HEUMANN PHARMA GMBH & CO (DE) 1986-11-05 EP disclosed