SCHEMBL9866302

SCHEMBL9866302

CC(C)(C)NCC(O)COc1ccc(-n2nc3c(cc2=O)COc2ccccc2-3)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.45
ADRB2 P07550 5/20 0.40
ADRB1 P08588 4/20 0.40
ADRB3 P13945 2/20 0.40
TSHR P16473 2/20 0.39
HTR1A P08908 1/20 0.39
SLC6A4 P31645 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
MEN1 O00255 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRA1A P35348 1/20 0.38
RECQL P46063 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867905 0.89 ADRB2 (0.44) CYP2D6ADRB2ADRB1ADRB3TSHR
SCHEMBL9867229 0.81 TOP1 (0.40)
SCHEMBL9865164 0.79 MAOB (0.37) CYP2D6TSHRHTR1ASLC6A4SIGMAR1
SCHEMBL9603116 0.79 CYP2D6 (0.41) CYP2D6ADRB2ADRB1ADRB3TSHR
SCHEMBL9865298 0.74 MCHR1 (0.43) CYP2D6TSHRHTR1ASLC6A4SIGMAR1
SCHEMBL9866651 0.70 ADRB2 (0.45) CYP2D6ADRB2ADRB1ADRB3TSHR
SCHEMBL9866045 0.69 THRB (0.34) MEN1KMT2A
SCHEMBL9602957 0.68 PTGS1 (0.42) CYP2D6ADRB2ADRB1ADRB3TSHR
SCHEMBL9865872 0.67 ADRB2 (0.44) ADRB2ADRB1ADRB3TSHRADRA1A
SCHEMBL11167444 0.67 MEN1 (0.53) CYP2D6ADRB2ADRB1ADRB3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5045541-A Immunodeficiency disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-09-03 US disclosed
EP-0351435-A1 FUSED PYRIDAZINE COMPOUNDS AND THEIR MEDICINAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-01-24 EP disclosed