SCHEMBL9866700

SCHEMBL9866700

CC(C)(C)OC(=O)N=C(N)N(CCCCCC(=O)Nc1cc(C(=O)NCCC(=O)O)cc([N+](=O)[O-])c1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.38
ITGA2 P17301 1/20 0.38
HDAC3 O15379 3/20 0.36
HDAC1 Q13547 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 4/20 0.35
LMNA P02545 4/20 0.35
MEN1 O00255 5/20 0.34
KMT2A Q03164 5/20 0.34
MAPT P10636 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 3/20 0.33
MITF O75030 1/20 0.33
XBP1 P17861 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9337501 0.82 HDAC1 (0.40) ITGB3ITGA2HDAC3HDAC1L3MBTL1
SCHEMBL9865729 0.80 CA1 (0.45) ITGB3ITGA2HDAC3HDAC1L3MBTL1
SCHEMBL9866871 0.80 CYP2C9 (0.43) HDAC3HDAC1L3MBTL1LMNAKMT2A
SCHEMBL9335656 0.76 HDAC1 (0.50) ITGB3ITGA2HDAC3HDAC1L3MBTL1
SCHEMBL9335641 0.75 LTA4H (0.37) HDAC1MEN1KMT2AHDAC2HDAC8
SCHEMBL9335626 0.75 HDAC1 (0.49) ITGB3ITGA2HDAC3HDAC1L3MBTL1
Formic Acid SCHEMBL9339472 0.73 HDAC1 (0.47) ITGB3ITGA2HDAC3HDAC1L3MBTL1
SCHEMBL9337513 0.73 CA1 (0.44) HDAC3HDAC1ALDH1A1LMNAMEN1
SCHEMBL9865333 0.70 CA1 (0.48) HDAC3HDAC1L3MBTL1MEN1KMT2A
SCHEMBL2905983 0.69 HDAC1 (0.33) HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5039805-A Novel benzoic and phenylacetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1991-08-13 US disclosed