SCHEMBL9335641

SCHEMBL9335641

CC(C)(C)OC(=O)/N=C(\N)N(CCCCC(=O)Nc1ccc(OCc2ccccc2)c(C(=O)NCCC(=O)O)c1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 4/20 0.37
C5AR1 P21730 7/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LRRK2 Q5S007 2/20 0.35
HDAC8 Q9BY41 1/20 0.35
P2RX4 Q99571 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866871 0.85 CYP2C9 (0.43) HDAC8KMT2AHDAC1HDAC2
SCHEMBL9864708 0.83 HDAC8 (0.40) LTA4HNPC1RAB9ATDP1LRRK2
SCHEMBL9337449 0.81 CA1 (0.47) LTA4HNPC1RAB9ATDP1LRRK2
SCHEMBL9337569 0.78 LTA4H (0.54) LTA4HNPC1RAB9ALRRK2HDAC8
SCHEMBL9335876 0.77 LTA4H (0.44) LTA4HNPC1RAB9ALRRK2HDAC8
SCHEMBL9866700 0.75 ITGB3 (0.38) HDAC8MEN1KMT2AHDAC1HDAC2
SCHEMBL9335827 0.74 CA1 (0.45) LTA4HLRRK2HDAC8MEN1KMT2A
SCHEMBL5487724 0.72 CHRNB2 (0.46)
SCHEMBL9866032 0.72 CA1 (0.50) LTA4HNPC1RAB9ATDP1LRRK2
SCHEMBL21408642 0.72 GFER (0.43) RAB9AHDAC8MEN1KMT2AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0372486-B1 Benzoic-acid phenylacetic-acid derivatives, their preparation and their use as medicines HOFFMANN LA ROCHE (CH) 1994-06-01 EP disclosed
US-5039805-A Novel benzoic and phenylacetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1991-08-13 US disclosed
EP-0372486-A2 Benzoic-acid phenylacetic-acid derivatives, their preparation and their use as medicines F. HOFFMANN-LA ROCHE AG (CH) 1990-06-13 EP disclosed