SCHEMBL986734

SCHEMBL986734

CCc1cc(C(=O)Cl)cc(CC)c1OC

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
TPMT P51580 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GLRA1 P23415 1/20 0.36
PTGS2 P35354 1/20 0.36
MAPK1 P28482 1/20 0.36
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10322938 0.84 HPGD (0.41) ALDH1A1KDM4EGAAMAPTHPGD
SCHEMBL1573216 0.82 TPMT (0.52) ALDH1A1KDM4ETPMTPTGS2
SCHEMBL10603556 0.80 PPARA (0.47) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL11672950 0.80 KDM4E (0.50) ALDH1A1KDM4EGAAMAPTHPGD
SCHEMBL2153655 0.79 HSP90AA1 (0.36) ALDH1A1GAATPMTGLRA1MAPT
SCHEMBL8473100 0.78 HMGCR (0.44) ALDH1A1KDM4EGAATPMTMEN1
SCHEMBL2154378 0.77 HSP90AA1 (0.35) ALDH1A1MEN1KMT2AGLRA1
SCHEMBL9549933 0.76 PTGS2 (0.46) ALDH1A1KDM4EMEN1KMT2APTGS2
SCHEMBL219096 0.75 TUBB4A (0.55) ALDH1A1KDM4ETPMTMEN1KMT2A
SCHEMBL4311603 0.75 TPMT (0.39) ALDH1A1KDM4EGAATPMTGLRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7875631-B2 e.g.1-(3,5-dichlorophenyl)-2-formyl-6-methoxy-1,2,3,4-tetrahydroisoquinoline; to prevent and/or treat cancer and other abnormal cell growth, and metabolic as well as blood vessel proliferate disorders, in which uncontrolled expression of insulin-like growth factor-1 receptor is observed ANALYTECON S.A. (CH) 2011-01-25 US disclosed
US-4024273-A Coronary vasodilator and anti-anginal compositions comprising substituted benzofurans and benzothiophenes and methods of producing coronary vasodilation and anti-anginal activity SMITHKLINE CORPORATION (US) 1977-05-17 US disclosed
US-3947470-A CORONARY VASODILATORS, TREATMENT OF ANGINA PECTORIS SMITHKLINE CORPORATION (US) 1976-03-30 US disclosed