SCHEMBL9867948

SCHEMBL9867948

CCOC(=O)CCNC(=O)Nc1ccncc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
NAMPT P43490 7/20 0.54
KMT2A Q03164 2/20 0.54
GAA P10253 1/20 0.54
PTPN7 P35236 1/20 0.51
MDM2 Q00987 1/20 0.50
RAB9A P51151 1/20 0.50
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
PPID Q08752 1/20 0.46
TAAR1 Q96RJ0 1/20 0.45
MAPT P10636 1/20 0.45
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27519540 0.85 ALDH1A1 (0.82) ALDH1A1NAMPTKMT2AGAAPTPN7
SCHEMBL10731132 0.82 TOP2A (0.52) ALDH1A1NAMPTKMT2AGAARAB9A
SCHEMBL14476963 0.81 BCHE (0.61) ALDH1A1NAMPTKMT2AGAARAB9A
SCHEMBL9937346 0.81 ALDH1A1 (0.59) ALDH1A1KMT2APTPN7RAB9AKDM4E
SCHEMBL12989329 0.80 KMT2A (0.64) ALDH1A1NAMPTKMT2AMDM2RAB9A
SCHEMBL23303452 0.79 NAAA (0.57) ALDH1A1KMT2ARAB9AKDM4ELMNA
SCHEMBL6915485 0.79 ALDH1A1 (0.60) ALDH1A1NAMPTKMT2AGAAPTPN7
SCHEMBL9868290 0.79 BCHE (0.62) NAMPTKMT2AMDM2RAB9AKEAP1
SCHEMBL1883394 0.77 PIK3CG (0.54) ALDH1A1KDM4ELMNAPPID
SCHEMBL11310806 0.77 NAMPT (0.65) ALDH1A1NAMPTKMT2AMDM2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997667-A Pyridinyl compounds of N-carbamoyl-N-thiocarbamoyl- or N-amidino-glycine or beta-alanine useful as sweetening agents UNIVERSITE CLAUDE BERNARD (FR) 1991-03-05 US disclosed
EP-0321369-A1 Heterocyclic sweeteners derived from N-carbamoyl-, N-thiocarbamoyl or N-amidino-glycine or beta-alanine UNIVERSITE CLAUDE BERNARD - LYON 1 (FR) 1989-06-21 EP disclosed