SCHEMBL9869424

SCHEMBL9869424

O=C(O)c1ccc(COc2ccccc2)nc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.54
GPBAR1 Q8TDU6 3/20 0.52
CYSLTR1 Q9Y271 8/20 0.51
CYSLTR2 Q9NS75 6/20 0.51
MRGPRX4 Q96LA9 1/20 0.47
ALDH1A1 P00352 2/20 0.46
NPC1 O15118 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
THPO P40225 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869319 0.79 POLB (0.41) GPBAR1ALDH1A1KDM4ELMNATP53
SCHEMBL9869721 0.77 TSHR (0.50) KCNH2GPBAR1CYSLTR1CYSLTR2ALDH1A1
SCHEMBL9870267 0.76 KDM4E (0.40) ALDH1A1NPC1KDM4ELMNATP53
SCHEMBL9869225 0.76 CYSLTR1 (0.39) KCNH2GPBAR1CYSLTR1CYSLTR2ALDH1A1
SCHEMBL11188667 0.74 MRGPRX4 (0.78) KCNH2GPBAR1CYSLTR1MRGPRX4KDM4E
SCHEMBL24834805 0.73 GABRP (0.47) ALDH1A1NPC1KDM4EMEN1CYP1A2
SCHEMBL1368181 0.73 TP53 (0.63) MRGPRX4ALDH1A1NPC1KDM4ETP53
SCHEMBL10664344 0.73 KDM4E (0.61) GPBAR1CYSLTR1CYSLTR2ALDH1A1NPC1
SCHEMBL7454590 0.72 GPBAR1 (0.74) GPBAR1CYSLTR1CYSLTR2ALDH1A1NPC1
SCHEMBL31568498 0.72 MRGPRX4 (0.53) GPBAR1CYSLTR1MRGPRX4ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997947-A Forming 6-substituted pyridine-2,3-dicarboxylic esters followed by reacting with aminoalkanecarboxylic acid amide; herbicides, plant growth regulators CIBA-GEIGY CORPORATION (US) 1991-03-05 US disclosed
EP-0296109-A2 Derivatives of 2-(imidazolin-2-yl)nicotinic acid CIBA-GEIGY AG (CH) 1988-12-21 EP disclosed