SCHEMBL9869721

SCHEMBL9869721

CCOC(=O)c1ccc(COc2ccccc2)nc1C(=O)OCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
MAPK10 P53779 1/20 0.50
SMN1; SMN2 Q16637 5/20 0.49
CYSLTR2 Q9NS75 3/20 0.47
CYSLTR1 Q9Y271 3/20 0.47
MEN1 O00255 1/20 0.47
HSP90AA1 P07900 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 3/20 0.47
GAA P10253 1/20 0.47
KCNH2 Q12809 1/20 0.46
MAPT P10636 4/20 0.46
MAOB P27338 1/20 0.46
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869056 0.82 CA12 (0.46) TSHRL3MBTL1CYP1A2ALDH1A1MAOB
SCHEMBL9869213 0.82 CA12 (0.46) TSHRCYP1A2ALDH1A1GAAMAOB
SCHEMBL9308690 0.80 TSHR (0.50) TSHRMEN1KMT2ACYP1A2ALDH1A1
SCHEMBL9869424 0.77 KCNH2 (0.54) TSHRSMN1; SMN2CYSLTR2CYSLTR1MEN1
SCHEMBL9784691 0.75 KDM4E (0.55) TSHRSMN1; SMN2KMT2AL3MBTL1ALDH1A1
SCHEMBL9308330 0.74 TSHR (0.53) TSHRMEN1KMT2ACYP1A2ALDH1A1
SCHEMBL14021543 0.72 GPBAR1 (0.70) CYSLTR2CYSLTR1GPBAR1
SCHEMBL6306356 0.71 TSHR (0.50) TSHRMEN1KMT2ACYP1A2ALDH1A1
SCHEMBL9900502 0.71 HPGDS (0.58) TSHRMAPK10SMN1; SMN2MEN1KMT2A
SCHEMBL28619313 0.71 TSHR (0.50) TSHRMAPK10SMN1; SMN2MEN1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997947-A Forming 6-substituted pyridine-2,3-dicarboxylic esters followed by reacting with aminoalkanecarboxylic acid amide; herbicides, plant growth regulators CIBA-GEIGY CORPORATION (US) 1991-03-05 US disclosed