SCHEMBL9870731

SCHEMBL9870731

Cc1nccc(-c2ccccc2)c1/C=C/CO

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.40
TACR1 P25103 2/20 0.38
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
GRM4 Q14833 1/20 0.36
IKBKB O14920 1/20 0.36
CHUK O15111 1/20 0.36
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
CSF1R P07333 1/20 0.36
RET P07949 1/20 0.36
IGF1R P08069 1/20 0.36
FGFR1 P11362 1/20 0.36
PRKACA P17612 1/20 0.36
FLT1 P17948 1/20 0.36
LTK P29376 1/20 0.36
GRK5 P34947 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870737 1.00 CHEK1 (0.40) CHEK1TACR1MKNK1MKNK2GRM4
SCHEMBL9871811 0.79 HCAR2 (0.43) CHEK1TACR1MKNK1MKNK2CDK8
SCHEMBL9871808 0.79 HCAR2 (0.43) CHEK1TACR1MKNK1MKNK2CDK8
SCHEMBL9871387 0.78 MEN1 (0.44) CHEK1TACR1MKNK1MKNK2GRM4
SCHEMBL9871401 0.78 MEN1 (0.44) CHEK1TACR1MKNK1MKNK2GRM4
SCHEMBL9871200 0.77 CHEK1 (0.42) CHEK1TACR1MKNK1MKNK2GRM4
SCHEMBL8846070 0.77 CHEK1 (0.42) CHEK1TACR1GRM4IKBKBCHUK
SCHEMBL18433892 0.74 CYP17A1 (0.43) CHEK1GRM4IKBKBCHUKDAPK3
SCHEMBL9871017 0.74 KMT2A (0.43) TACR1CDK8MEN1ALDH1A1KMT2A
SCHEMBL9871013 0.74 KMT2A (0.43) TACR1CDK8MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed