SCHEMBL9871687

SCHEMBL9871687

CCOC(=O)C1=C(C)NC=CC1c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1D Q01668 7/20 0.59
ADORA3 P0DMS8 3/20 0.52
DHFR P00374 1/20 0.50
KDM4E B2RXH2 3/20 0.49
GAA P10253 2/20 0.49
ALDH1A1 P00352 5/20 0.46
LMNA P02545 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
POLB P06746 1/20 0.45
ALOX12 P18054 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
XBP1 P17861 1/20 0.45
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10346121 0.83 KDM4E (0.58) CACNA1DADORA3DHFRKDM4EGAA
SCHEMBL5241525 0.76 CACNA1D (0.46) CACNA1DADORA3GAAALDH1A1LMNA
SCHEMBL6299988 0.75 KDM4E (0.51) ADORA3KDM4EGAAALDH1A1LMNA
SCHEMBL3027412 0.73 ADORA3 (0.89) CACNA1DADORA3DHFRKDM4EGAA
SCHEMBL9027650 0.71 GAA (0.42) CACNA1DADORA3DHFRKDM4EGAA
SCHEMBL29173863 0.70 ADORA3 (0.82) CACNA1DADORA3DHFRKDM4EGAA
SCHEMBL11799255 0.69 CACNA1D (0.60) CACNA1DADORA3DHFRKDM4EGAA
SCHEMBL11669396 0.69 ADORA3 (0.68) CACNA1DADORA3DHFRKDM4EGAA
SCHEMBL10684386 0.69 ADORA3 (0.75) CACNA1DADORA3DHFRKDM4EGAA
SCHEMBL20610477 0.69 ADORA3 (1.00) CACNA1DADORA3KDM4EGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed