SCHEMBL9871816

SCHEMBL9871816

O=C1OC(=O)c2nc3cc(O)c(O)cc3cc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB2 Q9UBS0 1/20 0.35
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
GLA P06280 2/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ALOX15 P16050 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
EGFR P00533 2/20 0.31
PDGFRB P09619 2/20 0.31
PDGFRA P16234 2/20 0.31
MAPT P10636 3/20 0.31
MCL1 Q07820 2/20 0.31
AKR1B1 P15121 2/20 0.31
HPGD P15428 2/20 0.31
CA12 O43570 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
BCHE P06276 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10516399 0.75 PDE3B (0.44) RPS6KB2KDM4EALDH1A1GLAPDGFRB
SCHEMBL310881 0.74 NPC1 (0.58) KDM4EALDH1A1GLANPC1RAB9A
SCHEMBL9117555 0.69 MEN1 (0.41) KDM4EALDH1A1GLANPC1RAB9A
SCHEMBL9672578 0.69 MCL1 (0.50) KDM4EALDH1A1ALOX15TDP1EGFR
SCHEMBL10402599 0.68 DYRK1A (0.42) KDM4EALDH1A1NPC1RAB9AALOX15
SCHEMBL9979779 0.66 EGFR (0.42) RPS6KB2KDM4EALDH1A1GLANPC1
SCHEMBL10415195 0.66 GRM2 (0.38) KDM4EALDH1A1NPC1RAB9AALOX15
SCHEMBL10651328 0.66 ALOX5 (0.35) RPS6KB2ALDH1A1NPC1RAB9AALOX15
SCHEMBL10473035 0.64 ALOX15 (0.34) KDM4EALDH1A1RAB9AALOX15TDP1
SCHEMBL8564561 0.64 ALOX15 (0.34) ALOX15TDP1TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037983-A 6,7-dihydroxyquinoxalines as intermediates to beta-lactam antibiotics E. R. SQUIBB & SONS, INC. (US) 1991-08-06 US disclosed
US-4904775-A Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics E. R. SQUIBB & SONS, INC. (US) 1990-02-27 US disclosed
EP-0342423-A2 Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics E.R. SQUIBB & SONS, INC. (US) 1989-11-23 EP disclosed
EP-0303286-A1 2-Oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines E.R. Squibb & Sons, Inc. (US) 1989-02-15 EP disclosed
US-4777252-A 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines E. R. SQUIBB & SONS, INC. (US) 1988-10-11 US disclosed