SCHEMBL9872541

SCHEMBL9872541

NC(=O)CCN1CCC(C(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.53
HTR2A P28223 5/20 0.50
HTR2C P28335 2/20 0.50
HTR7 P34969 2/20 0.50
PRCP P42785 1/20 0.45
HTR6 P50406 1/20 0.44
MEN1 O00255 1/20 0.43
CHRM2 P08172 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
DRD1 P21728 1/20 0.43
ADRA1A P35348 1/20 0.43
OPRM1 P35372 1/20 0.43
DRD3 P35462 1/20 0.43
KMT2A Q03164 1/20 0.43
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
CCR3 P51677 1/20 0.42
CACNA1B Q00975 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10567673 0.81 HTR2A (0.52) CYP2D6HTR2AHTR2CHTR7HTR6
SCHEMBL7330054 0.81 CYP2D6 (0.80) CYP2D6HTR2AMEN1CHRM2HTR1A
SCHEMBL9872721 0.79 CYP2D6 (0.47) CYP2D6HTR2AHTR2CHTR7OPRM1
SCHEMBL10459141 0.79 HTR2A (0.53) CYP2D6HTR2AHTR2CHTR7HTR6
SCHEMBL7640547 0.79 DRD2 (0.58) CYP2D6HTR2AHTR7PRCPHTR6
SCHEMBL11712337 0.79 SLC6A3 (0.50) CYP2D6KMT2AKCNH2CACNA1B
Oxalic Acid SCHEMBL10557086 0.78 CYP2D6 (0.53) CYP2D6HTR2AHTR2CHTR7MEN1
Hydrochloric Acid SCHEMBL7329135 0.78 HTR2A (0.63) CYP2D6HTR2AHTR2CHTR7HTR6
Hydrochloric Acid SCHEMBL7658850 0.78 DRD2 (0.57) CYP2D6HTR2AHTR7PRCPHTR6
SCHEMBL10556073 0.77 HRH3 (0.55) CYP2D6HTR2AHTR1ADRD1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4032642-A SEDATIVES, TRANQUILIZERS A. H. ROBINS COMPANY, INCORPORATED (US) 1977-06-28 US claimed
US-5057524-A Asthma, dermatitis A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US disclosed