SCHEMBL9872850

SCHEMBL9872850

Nc1nc(SCCC(=O)c2ccccc2)c2nc[nH]c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.45
KMT2A Q03164 3/20 0.45
MAPT P10636 3/20 0.45
CYP1A2 P05177 4/20 0.43
CYP3A4 P08684 4/20 0.43
CYP2C19 P33261 4/20 0.43
HSD17B10 Q99714 2/20 0.43
HPGD P15428 2/20 0.43
HIF1A Q16665 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
TOP2A P11388 1/20 0.43
NUDT1 P36639 1/20 0.43
ENPP1 P22413 1/20 0.43
MEN1 O00255 2/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
CTNNB1 P35222 2/20 0.40
WNT3A P56704 2/20 0.40
LMNA P02545 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14050054 0.88 CYP1A2 (0.53) ALDH1A1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL9872864 0.81 CYP1A2 (0.67) ALDH1A1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL13742763 0.80 CYP1A2 (0.64) ALDH1A1CYP1A2CYP3A4CYP2C19HSD17B10
SCHEMBL13742811 0.77 CYP2D6 (0.57) ALDH1A1CYP1A2CYP3A4CYP2C19HSD17B10
SCHEMBL1464157 0.77 CYP1A2 (0.69) ALDH1A1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL2115655 0.76 PIN1 (0.64) ALDH1A1CYP1A2CYP3A4CYP2C19HSD17B10
SCHEMBL8826177 0.74 SLC29A1 (0.47) ALDH1A1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL13742856 0.72 CYP1A2 (0.67) ALDH1A1KMT2AMAPTCYP1A2CYP3A4
SCHEMBL4845428 0.72 POLB (0.47) ALDH1A1HSD17B10HPGDENPP1SMN1; SMN2
SCHEMBL14028457 0.72 ALDH1A1 (0.65) ALDH1A1KMT2AMAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017701-A Process for the preparation of purine derivatives BEECHAM GROUP, P.L.C. (GB) 1991-05-21 US disclosed
EP-0352953-A2 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 1990-01-31 EP disclosed