SCHEMBL9872864

SCHEMBL9872864

Nc1nc(SCCC(=O)c2ccccc2)c2[nH]cnc2n1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.67
CYP3A4 P08684 5/20 0.67
CYP2C19 P33261 5/20 0.67
ALDH1A1 P00352 5/20 0.67
CYP2D6 P10635 4/20 0.67
CYP2C9 P11712 3/20 0.67
HPGD P15428 3/20 0.67
HIF1A Q16665 2/20 0.67
HSD17B10 Q99714 2/20 0.67
TOP2A P11388 1/20 0.67
NUDT1 P36639 1/20 0.67
PIN1 Q13526 2/20 0.61
POLB P06746 2/20 0.61
ENPP1 P22413 2/20 0.61
SMN1; SMN2 Q16637 3/20 0.57
LMNA P02545 4/20 0.53
HTT P42858 3/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
MAP3K5 Q99683 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24846433 0.88 CYP1A2 (0.79) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL9872850 0.81 ALDH1A1 (0.45) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL24846512 0.80 CYP1A2 (1.00) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL887207 0.79 ENPP1 (0.70) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL24846509 0.77 CYP1A2 (0.88) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL12920817 0.77 CYP1A2 (1.00) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL2115657 0.76 PIN1 (1.00) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL24846480 0.76 ENPP1 (1.00) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL24846382 0.76 ENPP1 (0.84) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6
SCHEMBL24846383 0.74 CYP1A2 (0.74) CYP1A2CYP3A4CYP2C19ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017701-A Process for the preparation of purine derivatives BEECHAM GROUP, P.L.C. (GB) 1991-05-21 US disclosed
EP-0352953-A2 Process for the preparation of purine derivatives BEECHAM GROUP PLC (GB) 1990-01-31 EP disclosed