SCHEMBL9873091

SCHEMBL9873091

COc1c(F)ccc(F)c1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
CA14 Q9ULX7 2/20 0.37
MEP1B Q16820 1/20 0.37
NFE2L2 Q16236 3/20 0.33
TDP1 Q9NUW8 1/20 0.33
ACHE P22303 1/20 0.33
PAX8 Q06710 1/20 0.33
KMT2A Q03164 1/20 0.33
PTGS2 P35354 1/20 0.33
POLB P06746 1/20 0.33
CA4 P22748 1/20 0.33
TUBB1 Q9H4B7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21437058 0.87 TUBB1 (0.36) KDM4EALDH1A1MAPK1SMN1; SMN2MEP1B
SCHEMBL1994314 0.85 MEP1B (0.41) KDM4EALDH1A1MAPK1SMN1; SMN2CA12
SCHEMBL23829848 0.84 ALDH1A1 (0.37) KDM4EALDH1A1MAPK1SMN1; SMN2MEP1B
SCHEMBL10209739 0.84 CA2 (0.43) KDM4EALDH1A1MAPK1SMN1; SMN2CA1
SCHEMBL14037359 0.83 KDM4E (0.36) KDM4EALDH1A1MAPK1SMN1; SMN2CA12
SCHEMBL475141 0.81 ALDH1A1 (0.46) KDM4EALDH1A1MAPK1SMN1; SMN2CA12
SCHEMBL7962496 0.81 PDE4A (0.39) KDM4EALDH1A1MAPK1SMN1; SMN2MEP1B
SCHEMBL23324806 0.81 KDM4E (0.35) KDM4EALDH1A1MAPK1SMN1; SMN2MEP1B
SCHEMBL23894376 0.81 HTR2A (0.38) KDM4EALDH1A1MAPK1SMN1; SMN2MEP1B
SCHEMBL746439 0.81 CA4 (0.39) KDM4EALDH1A1MAPK1SMN1; SMN2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037983-A 6,7-dihydroxyquinoxalines as intermediates to beta-lactam antibiotics E. R. SQUIBB & SONS, INC. (US) 1991-08-06 US disclosed
US-4904775-A Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics E. R. SQUIBB & SONS, INC. (US) 1990-02-27 US disclosed
EP-0342423-A2 Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics E.R. SQUIBB & SONS, INC. (US) 1989-11-23 EP disclosed