Bromide

Bromide

SCHEMBL9873579

Br.O=C1CCN(CC#Cc2ccccc2)CCC1Br

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 known ✓ P31645 1/20 0.42
SLC6A3 known ✓ Q01959 1/20 0.42
SIGMAR1 known ✓ Q99720 1/20 0.41
LMNA P02545 2/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.47
GRIN1 Q05586 5/20 0.46
GRIN2B Q13224 1/20 0.46
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
GRM5 P41594 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL548941 0.77 ACHE (0.54) HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL1916659 0.76 ACHE (0.56) HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL14485306 0.71 LMNA (0.81) LMNAMAPK1RAB9AGRIN1GRIN2B
Bromide SCHEMBL7286166 0.71 MCHR1 (0.51) LMNAMAPK1SLC6A4SLC6A3HTR2A
SCHEMBL5730065 0.70 LMNA (0.78) LMNAMAPK1RAB9AGRIN1GRIN2B
Valine SCHEMBL6436086 0.69 TACR1 (0.47) SIGMAR1
SCHEMBL5668453 0.69 HTR2A (0.54) GRIN1GRIN2BSLC6A4SLC6A3HTR2A
Hydrochloric Acid SCHEMBL5666575 0.68 HTR2A (0.53) GRIN1GRIN2BSLC6A4SLC6A3HTR2A
SCHEMBL3634873 0.67 LMNA (0.56) LMNAMAPK1RAB9AGRIN1GRIN2B
SCHEMBL3251635 0.67 LMNA (0.56) LMNAMAPK1RAB9AGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068325-A Dopaminergic systems as hypotensives, sedatives, antitussives and/or antiphlogistics KARL THOMAE GMBH (DE) 1991-11-26 US disclosed