SCHEMBL9874404

SCHEMBL9874404

Clc1ccc(C(Br)[CH]Br)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.42
MAPK1 P28482 2/20 0.42
HIF1A Q16665 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41
ADRB2 P07550 1/20 0.41
CYP2A6 P11509 1/20 0.40
CYP19A1 P11511 4/20 0.38
IDO1 P14902 3/20 0.38
TDO2 P48775 3/20 0.38
BRD4 O60885 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ALOX15 P16050 1/20 0.33
APEX1 P27695 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL118609 0.78 HSD17B10 (0.42) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL9147474 0.75 TSHR (0.41) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL1411248 0.74 TSHR (0.46) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL6190849 0.73 TSHR (0.50) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL1500533 0.73 TSHR (0.50) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL624797 0.69 ADRB2 (0.56) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL29013799 0.69 TSHR (0.46) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL29200286 0.69 TSHR (0.46) TSHRMAPK1HIF1ATDP1LMNA
SCHEMBL7008999 0.69 IDO1 (0.47) TSHRIDO1TDO2SLC6A4SLC6A3
SCHEMBL2091212 0.67 MAPK1 (0.50) TSHRMAPK1HIF1ATDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254078-B1 PYRAN DERIVATIVES BASF Aktiengesellschaft (DE) 1991-02-06 EP disclosed
EP-0254078-A1 Pyran derivatives BASF Aktiengesellschaft (DE) 1988-01-27 EP disclosed