SCHEMBL9874867

SCHEMBL9874867

CN(C)CCNc1c2c(nc3ccccc13)CCCC2=O

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PABPC1 P11940 1/20 0.71
EIF4H Q15056 1/20 0.71
HRH3 Q9Y5N1 3/20 0.66
RAD52 P43351 2/20 0.60
HRH2 P25021 1/20 0.57
HRH1 P35367 1/20 0.57
ACHE P22303 7/20 0.56
BCHE P06276 2/20 0.53
NPC1 O15118 1/20 0.51
POLB P06746 1/20 0.51
SLC2A1 P11166 1/20 0.51
APOBEC3A P31941 1/20 0.51
RAB9A P51151 1/20 0.51
KMT2A Q03164 1/20 0.51
APOBEC3G Q9HC16 1/20 0.51
TERT O14746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9875611 0.87 BCHE (0.53) PABPC1EIF4HRAD52ACHEBCHE
SCHEMBL9875231 0.83 BCHE (0.64) ACHEBCHEKMT2A
Hydrochloric Acid SCHEMBL31087706 0.82 PABPC1 (0.97) PABPC1EIF4HHRH3RAD52HRH2
SCHEMBL8984077 0.81 KMT2A (0.67) RAD52ACHEBCHEPOLBKMT2A
SCHEMBL9875385 0.80 KDM4E (0.54) PABPC1EIF4HACHEBCHEPOLB
SCHEMBL9874141 0.80 BCHE (0.54) ACHEBCHESLC2A1
SCHEMBL9874160 0.80 BCHE (0.54) ACHEBCHESLC2A1
SCHEMBL9875000 0.78 KDM4E (0.57) RAD52ACHEBCHEPOLBKMT2A
SCHEMBL9874947 0.78 KDM4E (0.51) PABPC1EIF4HACHEBCHEKMT2A
SCHEMBL9736923 0.78 PABPC1 (0.69) PABPC1EIF4HHRH3RAD52HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4695573-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US claimed
EP-2681554-B1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON DICKINSON CO (US) 2017-08-09 EP disclosed
US-9459187-B2 Blood collection device containing lysophospholipase inhibitor BECTON, DICKINSON AND COMPANY (US) 2016-10-04 US disclosed
US-20140030754-A1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON, DICKINSON AND COMPANY (US) 2014-01-30 US disclosed
US-20130209985-A1 SAMPLE COLLECTION DEVICES WITH BLOOD STABILIZING AGENTS BECTON, DICKINSON AND COMPANY 2013-08-15 US disclosed
WO-2012121998-A1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON, DICKINSON AND COMPANY (US) 2012-09-13 WO disclosed
EP-0179383-B1 9-AMINO-1,2,3,4-TETRAHYDROACRIDIN-1-OL AND RELATED COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-05-29 EP disclosed
US-4839364-A ALZHEIMER*S DISEASE; CHOLINESTERASE INHIBITORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-06-13 US disclosed
US-4835275-A Method of preparing 9-amino-1,2,3,4,-tetrahydroacridin-1-ones and related compounds HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-05-30 US disclosed
US-4754050-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-06-28 US disclosed
US-4695573-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US disclosed
EP-0179383-A2 9-Amino-1,2,3,4-tetrahydroacridin-1-ol and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-04-30 EP disclosed