SCHEMBL9875274

SCHEMBL9875274

Nc1c2c(nc3ccc([N+](=O)[O-])cc13)CCCC2=O

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACHE P22303 15/20 0.67
KDM4E B2RXH2 1/20 0.52
BCHE P06276 7/20 0.49
APP P05067 2/20 0.49
TYMS P04818 1/20 0.42
GRIN1 Q05586 5/20 0.42
GRIN2A Q12879 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27995132 0.84 ACHE (0.53) ACHEKDM4EBCHEAPPTYMS
SCHEMBL9874888 0.82 ACHE (0.54) ACHEBCHEAPP
SCHEMBL9874322 0.81 ACHE (0.60) ACHEKDM4EBCHEGRIN1GRIN2A
SCHEMBL5988415 0.81 ACHE (1.00) ACHEBCHEAPPGRIN1GRIN2A
SCHEMBL9068077 0.79 ACHE (0.66) ACHEKDM4EBCHEGRIN1GRIN2A
SCHEMBL10848027 0.79 ACHE (0.66) ACHEKDM4EBCHEAPPGRIN1
SCHEMBL9873371 0.79 ACHE (0.68) ACHEKDM4EBCHEGRIN1GRIN2A
SCHEMBL10847043 0.79 ACHE (0.62) ACHEKDM4EBCHEGRIN1GRIN2A
SCHEMBL9736799 0.79 ACHE (0.69) ACHEBCHEAPP
SCHEMBL10845002 0.76 KDM4E (0.53) ACHEKDM4EBCHEGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4631286-A MEMORY ENHANCERS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-12-23 US claimed
EP-2681554-B1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON DICKINSON CO (US) 2017-08-09 EP disclosed
US-9459187-B2 Blood collection device containing lysophospholipase inhibitor BECTON, DICKINSON AND COMPANY (US) 2016-10-04 US disclosed
US-20140030754-A1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON, DICKINSON AND COMPANY (US) 2014-01-30 US disclosed
US-20130209985-A1 SAMPLE COLLECTION DEVICES WITH BLOOD STABILIZING AGENTS BECTON, DICKINSON AND COMPANY 2013-08-15 US disclosed
EP-0179383-B1 9-AMINO-1,2,3,4-TETRAHYDROACRIDIN-1-OL AND RELATED COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-05-29 EP disclosed
US-4839364-A ALZHEIMER*S DISEASE; CHOLINESTERASE INHIBITORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-06-13 US disclosed
US-4835275-A Method of preparing 9-amino-1,2,3,4,-tetrahydroacridin-1-ones and related compounds HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-05-30 US disclosed
US-4754050-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-06-28 US disclosed
US-4695573-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US disclosed
US-4631286-A MEMORY ENHANCERS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-12-23 US disclosed
EP-0179383-A2 9-Amino-1,2,3,4-tetrahydroacridin-1-ol and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-04-30 EP disclosed