SCHEMBL9876130

SCHEMBL9876130

C=C1CCc2nc3ccccc3c(N)c2C1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.55
ACHE P22303 10/20 0.51
BCHE P06276 6/20 0.51
HSD17B10 Q99714 6/20 0.50
ALDH1A1 P00352 6/20 0.50
GLA P06280 3/20 0.50
HPGD P15428 3/20 0.50
GAA P10253 2/20 0.50
TSHR P16473 5/20 0.48
CYP1A2 P05177 3/20 0.48
KCNH2 Q12809 3/20 0.48
CYP2D6 P10635 2/20 0.48
CHRM2 P08172 2/20 0.48
ADRA2A P08913 2/20 0.48
ADORA3 P0DMS8 2/20 0.48
CHRM1 P11229 2/20 0.48
SLC6A2 P23975 2/20 0.48
OPRM1 P35372 2/20 0.48
CACNB4 O00305 1/20 0.48
CACNA1A O00555 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9875563 0.81 KDM4E (0.68) KDM4EACHEBCHEHSD17B10ALDH1A1
SCHEMBL10851259 0.79 KDM4E (0.55) KDM4EACHEBCHEHSD17B10ALDH1A1
SCHEMBL4495989 0.76 KDM4E (0.82) KDM4EACHEBCHEHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL8984092 0.75 KDM4E (0.80) KDM4EACHEBCHEHSD17B10ALDH1A1
SCHEMBL7272513 0.71 HSD17B10 (0.54) KDM4EACHEBCHEHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL7271547 0.70 MEN1 (0.56) KDM4EACHEBCHEHSD17B10ALDH1A1
SCHEMBL10850801 0.69 ACHE (0.52) KDM4EACHEBCHEHSD17B10ALDH1A1
SCHEMBL8543201 0.68 ACHE (0.51) KDM4EACHEBCHEHSD17B10ALDH1A1
SCHEMBL9587655 0.68 ACHE (0.51) KDM4EACHEBCHEHSD17B10ALDH1A1
SCHEMBL8542085 0.67 ACHE (0.50) KDM4EACHEBCHEHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4631286-A MEMORY ENHANCERS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-12-23 US claimed
EP-2681554-B1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON DICKINSON CO (US) 2017-08-09 EP disclosed
US-9459187-B2 Blood collection device containing lysophospholipase inhibitor BECTON, DICKINSON AND COMPANY (US) 2016-10-04 US disclosed
US-20140030754-A1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON, DICKINSON AND COMPANY (US) 2014-01-30 US disclosed
US-20130209985-A1 SAMPLE COLLECTION DEVICES WITH BLOOD STABILIZING AGENTS BECTON, DICKINSON AND COMPANY 2013-08-15 US disclosed
EP-0179383-B1 9-AMINO-1,2,3,4-TETRAHYDROACRIDIN-1-OL AND RELATED COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-05-29 EP disclosed
US-4839364-A ALZHEIMER*S DISEASE; CHOLINESTERASE INHIBITORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-06-13 US disclosed
US-4835275-A Method of preparing 9-amino-1,2,3,4,-tetrahydroacridin-1-ones and related compounds HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-05-30 US disclosed
US-4754050-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-06-28 US disclosed
US-4695573-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US disclosed
US-4631286-A MEMORY ENHANCERS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-12-23 US disclosed
EP-0179383-A2 9-Amino-1,2,3,4-tetrahydroacridin-1-ol and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-04-30 EP disclosed