SCHEMBL987621

SCHEMBL987621

O=C(CNN1CCCC1)N1CCC[C@H]1B(O)O

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 18/20 0.66
DPP7 Q9UHL4 11/20 0.66
FAP Q12884 19/20 0.64
PREP P48147 7/20 0.64
DPP8 Q6V1X1 2/20 0.59
DPP9 Q86TI2 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3641383 1.00 DPP4 (0.66) DPP4DPP7FAPPREPDPP8
SCHEMBL8286531 0.81 FAP (0.72) DPP4DPP7FAPPREPDPP8
SCHEMBL3204887 0.79 DPP4 (1.00) DPP4DPP7FAPPREPDPP8
SCHEMBL8243717 0.78 FAP (1.00) DPP4DPP7FAPPREPDPP8
SCHEMBL8285595 0.78 FAP (0.72) DPP4DPP7FAPPREPDPP8
SCHEMBL8285586 0.78 DPP4 (1.00) DPP4DPP7FAPPREPDPP8
SCHEMBL29362440 0.78 FAP (1.00) DPP4DPP7FAPPREPDPP8
SCHEMBL7901012 0.78 DPP4 (1.00) DPP4DPP7FAPPREPDPP8
SCHEMBL8244087 0.78 FAP (1.00) DPP4DPP7FAPPREPDPP8
SCHEMBL8244085 0.78 DPP4 (0.66) DPP4DPP7FAPPREPDPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005929-A1 PIPERIDINE DERIVATIVE AND ITS USE FOR THE TREATMENT OF DIABETS AND OBESITY ARENA PHARMACEUTICALS, INC. (US) 2011-01-13 WO disclosed
US-7786312-B2 Methods of preparing heterocyclic boronic acids and derivatives thereof PHENOMIX CORPORATION (US) 2010-08-31 US disclosed
US-20080300413-A1 Methods of Preparing Hetercyclic Boronic Acids and Derivatives Thereof SINO-MED INTERNATIONAL ALLIANCE, INC. 2008-12-04 US disclosed
EP-1919485-A1 METHODS OF PREPARING HETERCYCLIC BORONIC ACIDS AND DERIVATIVES THEREOF Phenomix Corporation (US) 2008-05-14 EP disclosed
WO-2007016356-A1 METHODS OF PREPARING HETERCYCLIC BORONIC ACIDS AND DERIVATIVES THEREOF PHENOMIX CORPORATION (US) 2007-02-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080300413-A1 Methods of Preparing Hetercyclic Boronic Acids and Derivatives Thereof HLCS, NISCH, BTD DPP4 1428/4885DPP7 1927/4885FAP 922/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.