SCHEMBL9876216

SCHEMBL9876216

CC1(C)C=Cc2cc(C#N)c(N)cc2O1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
CYP3A4 P08684 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
CA7 P43166 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CA9 Q16790 1/20 0.40
CA13 Q8N1Q1 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TLR3 O15455 1/20 0.34
ODC1 P11926 1/20 0.34
ABCB1 P08183 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8069868 0.84 ALDH1A1 (0.42) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL8069838 0.81 ALDH1A1 (0.42) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL8882171 0.79 ODC1 (0.46) ODC1
SCHEMBL11158278 0.77 TLR3 (0.47) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL31254002 0.76 ALDH1A1 (0.45) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL13476117 0.74 TLR3 (0.47) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL30523681 0.71 CA12 (0.46) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL20766474 0.71 ODC1 (0.44) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL30065854 0.71 ODC1 (0.44) ALDH1A1HPGDCYP3A4TDP1KDM4E
SCHEMBL506743 0.71 CA12 (0.46) ALDH1A1HPGDCYP3A4TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5071871-A Pharmaceutically useful benzo(β)pyranes and pyranopyridines SANDOZ LTD. (CH) 1991-12-10 US disclosed
EP-0028449-B1 CHROMANOL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND A PHARMACEUTICAL COMPOSITION COMPRISING THEM BEECHAM GROUP PLC (GB) 1983-07-20 EP disclosed
US-4366163-A Anti-hypertensive chromanol derivatives BEECHAM GROUP LIMITED (GB) 1982-12-28 US disclosed
US-4353906-A Chromanol derivatives and their use for treating hypertension BEECHAM GROUP LIMITED (GB) 1982-10-12 US disclosed
EP-0033613-A1 Chromanol derivatives, a process for their preparation and compositions containing them BEECHAM GROUP PLC (GB) 1981-08-12 EP disclosed
EP-0028449-A1 Chromanol derivatives, a process for their preparation and a pharmaceutical composition comprising them BEECHAM GROUP PLC (GB) 1981-05-13 EP disclosed