SCHEMBL9877022

SCHEMBL9877022

CCOC(=O)CCN(C(N)=S)c1ccc2cn[nH]c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 1/20 0.38
INSR P06213 1/20 0.38
IGF1R P08069 1/20 0.38
MAPT P10636 6/20 0.37
ALDH1A1 P00352 6/20 0.37
NEK2 P51955 1/20 0.37
KDM4E B2RXH2 7/20 0.37
DHODH Q02127 1/20 0.37
QPCT Q16769 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
FGFR1 P11362 2/20 0.36
FGFR2 P21802 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868330 0.76 SMN1; SMN2 (0.40) SMN1; SMN2HPGDMAPTALDH1A1KDM4E
SCHEMBL9877025 0.70 RECQL (0.67) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL562951 0.68 MEN1 (0.65) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL11954287 0.67 CYP1A2 (0.44) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL731312 0.67 MEN1 (0.64) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL25231993 0.66 PDE3B (0.55) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL30427608 0.66 PDE3B (0.55) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL11954389 0.66 MEN1 (0.47) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5823007 0.66 MAPT (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9867945 0.64 SMN1; SMN2 (0.50) SMN1; SMN2CYP1A2HPGDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997667-A Pyridinyl compounds of N-carbamoyl-N-thiocarbamoyl- or N-amidino-glycine or beta-alanine useful as sweetening agents UNIVERSITE CLAUDE BERNARD (FR) 1991-03-05 US disclosed
EP-0321369-A1 Heterocyclic sweeteners derived from N-carbamoyl-, N-thiocarbamoyl or N-amidino-glycine or beta-alanine UNIVERSITE CLAUDE BERNARD - LYON 1 (FR) 1989-06-21 EP disclosed