SCHEMBL9877341

SCHEMBL9877341

COc1cccc2c1C(=O)c1c(OC)cc(CNCCO)cc1C2=O

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.48
PIM1 P11309 1/20 0.48
ELANE P08246 7/20 0.47
CD274 Q9NZQ7 2/20 0.46
PDCD1 Q15116 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CTSG P08311 1/20 0.44
KDM4E B2RXH2 1/20 0.43
POLB P06746 1/20 0.43
PDCD1LG2 Q9BQ51 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878187 0.88 EGFR (0.45) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL9877590 0.86 ELANE (0.51) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL9877882 0.85 ALDH1A1 (0.60) ELANECD274PDCD1MEN1KMT2A
SCHEMBL8996370 0.83 EGFR (0.58) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL9878218 0.79 EGFR (0.54) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL9879835 0.79 EGFR (0.48) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL28440561 0.78 EGFR (0.52) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL15413506 0.78 ELANE (0.53) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL3272451 0.78 MEN1 (0.68) ELANEMEN1KMT2ACTSGKDM4E
SCHEMBL11432952 0.75 MEN1 (0.72) EGFRPIM1ELANEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4966918-A ANTICARCINOGENIC AGENTS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-10-30 US claimed
WO-1990008759-A1 DERIVATIVES OF CHRYSOPHANOL SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-08-09 WO claimed
US-5053431-A Antitumor-anticarcinogenic agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1991-10-01 US disclosed
US-4966918-A ANTICARCINOGENIC AGENTS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-10-30 US disclosed
WO-1990008759-A1 DERIVATIVES OF CHRYSOPHANOL SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-08-09 WO disclosed