SCHEMBL9877882

SCHEMBL9877882

COc1cc(OC)c2c(c1)C(=O)c1cc(CNCCO)cc(OC)c1C2=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 2/20 0.60
ELANE P08246 4/20 0.49
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
RECQL P46063 1/20 0.40
GLA P06280 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
BLM P54132 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9877592 0.88 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4ELANEMEN1
SCHEMBL9878587 0.86 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP3A4ELANEMEN1
SCHEMBL9877341 0.85 EGFR (0.48) ELANEMEN1KMT2AKDM4EPOLB
SCHEMBL9877371 0.85 ELANE (0.56) ALDH1A1CYP1A2CYP3A4ELANEMEN1
SCHEMBL9878499 0.78 ALDH1A1 (0.75) ALDH1A1CYP1A2CYP3A4ELANEKDM4E
SCHEMBL9879947 0.78 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4ELANEKDM4E
SCHEMBL16226679 0.78 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP3A4ELANEKDM4E
SCHEMBL16225747 0.76 ALDH1A1 (0.61) ALDH1A1CYP1A2CYP3A4ELANEMEN1
SCHEMBL27820157 0.75 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4ELANEKDM4E
SCHEMBL28005845 0.75 ALDH1A1 (0.69) ALDH1A1CYP1A2CYP3A4ELANEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5053431-A Antitumor-anticarcinogenic agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1991-10-01 US disclosed
US-4966918-A ANTICARCINOGENIC AGENTS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-10-30 US disclosed
WO-1990008759-A1 DERIVATIVES OF CHRYSOPHANOL SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-08-09 WO disclosed