SCHEMBL9877648

SCHEMBL9877648

CCC(C(=O)c1cccnc1)c1ccc(Cl)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
LMNA P02545 3/20 0.48
KDM4E B2RXH2 1/20 0.48
PKM P14618 1/20 0.48
P2RX7 Q99572 1/20 0.46
KMT2A Q03164 3/20 0.45
RAB9A P51151 2/20 0.45
MEN1 O00255 2/20 0.45
NPC1 O15118 1/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
MAPT P10636 2/20 0.44
POLB P06746 1/20 0.44
KCNMA1 Q12791 1/20 0.43
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878025 0.90 ALDH1A1 (0.46) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL11096738 0.86 ALDH1A1 (0.45) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL10528004 0.86 ALDH1A1 (0.45) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL6204706 0.85 NPC1 (0.46) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL11122644 0.85 ALDH1A1 (0.46) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL11094696 0.84 ALDH1A1 (0.48) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL9877329 0.84 ALDH1A1 (0.46) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL11094694 0.84 ALDH1A1 (0.48) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL6202785 0.84 NPC1 (0.46) ALDH1A1LMNAKDM4EPKMKMT2A
SCHEMBL10448844 0.84 ALDH1A1 (0.48) ALDH1A1LMNAKDM4EPKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5036074-A In agriculture and horticulture CIBA-GEIGY CORPORATION (US) 1991-07-30 US disclosed
EP-0385267-A2 Pyridine derivatives, their preparation and their use as fungicides CIBA-GEIGY AG (CH) 1990-09-05 EP disclosed
US-4753947-A Certain fungicidal alphabenzyl-3-pyridylmethanol, the corresponding chloro derivatives thereof or the N-oxides thereof HOFFMANN-LA ROCHE INC. (US) 1988-06-28 US disclosed
EP-0137456-B1 DERIVATIVES OF PYRIDINE, PYRAZINE AND PYRIMIDINE AND THEIR USE AS FUNGICIDAL AGENTS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1988-02-10 EP disclosed
US-4678790-A AGRICULTURE HORTICULTURE HOFFMAN-LA ROCHE INC. (US) 1987-07-07 US disclosed
EP-0074018-B1 PYRIDINE AND PYRAZINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THESE COMPOUNDS, FUNGICIDES CONTAINING THESE COMPOUNDS AS ACTIVE SUBSTANCES, USE OF THESE COMPOUNDS OR FUNGICIDES TO COMBAT FUNGI IN AGRICULTURE AND IN HORTICULTURE, AND KETONES AND FUNGICIDES CONTAINING THEM F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1986-09-24 EP disclosed
US-4556661-A FUNGICIDES HOFFMANN-LA ROCHE INC. (US) 1985-12-03 US disclosed
EP-0137456-A1 Derivatives of pyridine, pyrazine and pyrimidine and their use as fungicidal agents F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-04-17 EP disclosed
EP-0062238-B1 1,3-DIOXOLANE DERIVATIVES, THEIR PREPARATION, FUNGICIDAL AGENTS CONTAINING THOSE COMPOUNDS AS ACTIVE AGENTS AND USE OF SUCH COMPOUNDS OR AGENTS IN COMBATING FUNGI IN AGRICULTURE AND IN GARDENING F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1985-01-30 EP disclosed
US-4380544-A 1,3-Dioxolane compounds and their use as fungicides HOFFMANN-LA ROCHE INC. (US) 1983-04-19 US disclosed
EP-0074018-A2 Pyridine and pyrazine derivatives, process for the preparation of these compounds, fungicides containing these compounds as active substances, use of these compounds or fungicides to combat fungi in agriculture and in horticulture, and ketones and fungicides containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-03-16 EP disclosed
EP-0062238-A1 1,3-Dioxolane derivatives, their preparation, fungicidal agents containing those compounds as active agents and use of such compounds or agents in combating fungi in agriculture and in gardening F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-10-13 EP disclosed