SCHEMBL6202785

SCHEMBL6202785

O=C(c1cccnc1)C(Cc1ccccc1)c1ccc(Cl)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.46
ALDH1A1 P00352 3/20 0.46
LMNA P02545 3/20 0.46
KDM4E B2RXH2 1/20 0.46
PKM P14618 1/20 0.46
ECE1 P42892 1/20 0.45
RAB9A P51151 3/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
HDAC8 Q9BY41 1/20 0.43
TSHR P16473 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204706 0.94 NPC1 (0.46) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL6200990 0.86 MAPT (0.44) ALDH1A1LMNAKDM4EPKMRAB9A
SCHEMBL9877648 0.84 ALDH1A1 (0.48) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL9878025 0.82 ALDH1A1 (0.46) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL6199987 0.82 RAB9A (0.43) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL6203751 0.82 MAPK1 (0.46) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL11094696 0.81 ALDH1A1 (0.48) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL11094694 0.81 ALDH1A1 (0.48) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL9877329 0.81 ALDH1A1 (0.46) NPC1ALDH1A1LMNAKDM4EPKM
SCHEMBL10448844 0.81 ALDH1A1 (0.48) NPC1ALDH1A1LMNAKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed
EP-0117485-A2 Pyridine, pyrazine and pyrimidine derivatives and their use as fungicides F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-09-05 EP disclosed