SCHEMBL9878956

SCHEMBL9878956

CSc1nc(=O)c2c([nH]1)CCCC2

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
HPGD P15428 2/20 0.50
SMN1; SMN2 Q16637 3/20 0.41
ALOX15 P16050 1/20 0.41
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.37
MAPT P10636 4/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
HIF1A Q16665 1/20 0.37
CDKN1A P38936 1/20 0.36
HAVCR2 Q8TDQ0 1/20 0.36
PARP1 P09874 1/20 0.35
KMT2A Q03164 1/20 0.35
ELANE P08246 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878600 0.79 MEN1 (0.45) ALDH1A1HPGDSMN1; SMN2GAAMAPT
SCHEMBL14942690 0.76 HAVCR2 (0.56) ALDH1A1SMN1; SMN2ALOX15TSHRMAPT
SCHEMBL14029138 0.75 SMN1; SMN2 (0.41) ALDH1A1HPGDSMN1; SMN2ALOX15TSHR
SCHEMBL1702021 0.73 ALDH1A1 (0.41) ALDH1A1HPGDSMN1; SMN2GAAMAPT
SCHEMBL10568178 0.72 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2ALOX15TSHRMAPT
SCHEMBL9878958 0.71 HPGD (0.57) ALDH1A1HPGDGAAMAPTLMNA
SCHEMBL3536004 0.70 MAPT (0.65) ALDH1A1HPGDSMN1; SMN2MAPTLMNA
SCHEMBL7992628 0.70 ALDH1A1 (0.67) ALDH1A1HPGDSMN1; SMN2TSHRMAPT
SCHEMBL9880004 0.70 ALDH1A1 (0.36) ALDH1A1HPGDSMN1; SMN2MAPTHTT
SCHEMBL3583064 0.70 MAPT (0.64) ALDH1A1HPGDSMN1; SMN2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018887-A1 DIAMINOPYRIMIDINE COMPOUNDS SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1991-12-12 WO disclosed