SCHEMBL9878971

SCHEMBL9878971

Cc1[nH]c(C)c(-c2ccc(-c3ccc(F)cc3)cc2)c(=O)c1Cl.Cc1cc(=O)c(-c2ccc(Oc3ccccc3)cc2)c(C)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.47
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
BLM P54132 1/20 0.37
GSTP1 P09211 1/20 0.36
SCN9A Q15858 4/20 0.35
DHODH Q02127 2/20 0.34
PARP1 P09874 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
TYMP P19971 1/20 0.34
BCL2L1 Q07817 1/20 0.34
MCL1 Q07820 1/20 0.34
GPR84 Q9NQS5 1/20 0.33
CHEK2 O96017 1/20 0.33
PTGS2 P35354 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9265637 0.83 GSTP1 (0.51) SLC2A1CYP1A2POLBCYP3A4CYP2C9
SCHEMBL9266330 0.79 TYMP (0.50) SLC2A1TYMPPTGS2MEN1KMT2A
SCHEMBL9262778 0.78 TYMP (0.51) SLC2A1TYMPPTGS2MEN1KMT2A
SCHEMBL9259612 0.78 KEAP1 (0.47) KEAP1NFE2L2TYMPPTGS2MEN1
SCHEMBL9268241 0.77 SLC2A1 (0.63) SLC2A1CYP1A2POLBCYP3A4CYP2C9
SCHEMBL9455077 0.76 KEAP1 (0.49) KEAP1NFE2L2TYMPPTGS2MEN1
SCHEMBL9270359 0.75 SLC2A1 (0.78) SLC2A1CYP1A2POLBCYP3A4CYP2C9
SCHEMBL4469241 0.74 SLC2A1 (0.51) SLC2A1SCN9ACHEK2
SCHEMBL9266167 0.74 SLC2A1 (0.51) SLC2A1CYP1A2POLBCYP3A4CYP2C9
SCHEMBL9269889 0.74 PDGFRA (0.49) CYP1A2POLBPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991013873-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-19 WO disclosed