SCHEMBL9259612

SCHEMBL9259612

Cc1cc(=O)c(-c2ccc(-c3ccc(F)cc3)cc2)c(C)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
TNKS2 Q9H2K2 1/20 0.44
PTGS2 P35354 2/20 0.43
TYMP P19971 1/20 0.40
GCGR P47871 1/20 0.40
MAPK14 Q16539 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
SLC11A2 P49281 1/20 0.38
CTSV O60911 1/20 0.37
CTSL P07711 1/20 0.37
PGR P06401 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9455077 0.98 KEAP1 (0.49) KEAP1NFE2L2TNKS2PTGS2TYMP
SCHEMBL9269889 0.84 PDGFRA (0.49) TNKS2PTGS2SMN1; SMN2KDM4EPGR
SCHEMBL9455121 0.84 ALDH1A1 (0.46) PTGS2ADORA1MEN1KMT2ASMN1; SMN2
SCHEMBL5100169 0.83 SLC2A1 (0.48) PTGS2MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL9269940 0.81 SLC2A1 (0.49) PTGS2MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL3398595 0.81 LMNA (0.49) KEAP1NFE2L2TNKS2PTGS2ADORA1
SCHEMBL9422608 0.80 PDGFRA (0.51) PTGS2SMN1; SMN2KDM4EMAPT
SCHEMBL9454944 0.80 MAPT (0.53) TNKS2PTGS2SLC11A2MAPT
SCHEMBL9454898 0.78 ALDH1A1 (0.51) PTGS2SMN1; SMN2KDM4EMAPT
SCHEMBL9878971 0.78 SLC2A1 (0.47) KEAP1NFE2L2PTGS2TYMPMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403934-A Heterocyclic compounds BURROUGHS WELLCOME CO. (US) 1995-04-04 US disclosed
WO-1991013873-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-19 WO disclosed