SCHEMBL9890769

SCHEMBL9890769

CNC(=O)Cc1ccc(Cl)cc1-c1cccc(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 5/20 0.50
CHRM3 P20309 2/20 0.50
PDE4B Q07343 1/20 0.46
VEGFA P15692 1/20 0.44
FLT1 P17948 1/20 0.44
EGLN1 Q9GZT9 1/20 0.44
EGLN3 Q9H6Z9 1/20 0.44
PDE4D Q08499 1/20 0.43
NUDT1 P36639 1/20 0.43
GCGR P47871 1/20 0.42
KCNJ5 P48544 1/20 0.42
KCNJ3 P48549 1/20 0.42
SHMT1 P34896 1/20 0.41
SHMT2 P34897 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
RORC P51449 2/20 0.41
SOS1 Q07889 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2393525 0.90 PTGDR2 (0.47) CHRM1CHRM3SHMT1SHMT2
SCHEMBL9890716 0.89 CHRM1 (0.62) CHRM1CHRM3PDE4BVEGFAFLT1
SCHEMBL9890669 0.82 SUCNR1 (0.47) CHRM1CHRM3GCGRSHMT1SHMT2
SCHEMBL9890768 0.81 PDE4B (0.45) CHRM1CHRM3PDE4BPDE4DNUDT1
SCHEMBL9890728 0.78 FFAR1 (0.46) CHRM1CHRM3SHMT1SHMT2
SCHEMBL2395234 0.78 CNR1 (0.43) CHRM1CHRM3GCGR
SCHEMBL9890765 0.77 SMN1; SMN2 (0.43) CHRM3
SCHEMBL4247795 0.77 ERCC1 (0.56)
SCHEMBL9890789 0.76 CHRM3 (0.40) CHRM1CHRM3
SCHEMBL9926464 0.75 P2RX7 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US disclosed
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-06-07 US disclosed
EP-2374790-A1 BIPHENYLACETAMIDE DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2011-10-12 EP disclosed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US disclosed
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142771-A1 BIPHENYLACETAMIDE DERIVATIVE HRH3, KCNH3, BRPF3 CHRM1 340/4885CHRM3 298/4885PDE4B 3015/4885
US-20110224304-A1 BIPHENYLACETAMIDE DERIVATIVE HRH3, KCNH3, BRPF3 CHRM1 340/4885CHRM3 298/4885PDE4B 3015/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.