SCHEMBL9892862

SCHEMBL9892862

CC(C)(C)OC(=O)N1CC[C@H]1C(=O)Nc1nnc(-c2ccccc2)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 6/20 0.47
NPC1 O15118 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.42
PRMT5 O14744 1/20 0.41
UCHL1 P09936 3/20 0.40
HDAC8 Q9BY41 1/20 0.40
BUB1 O43683 1/20 0.40
HPGDS O60760 1/20 0.39
JAK2 O60674 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN6 P29350 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7075835 0.79 NPC1 (0.65) USP30NPC1MEN1KMT2ALMNA
SCHEMBL7075840 0.79 NPC1 (0.65) USP30NPC1MEN1KMT2ALMNA
SCHEMBL16054075 0.78 HPGDS (0.45) USP30MEN1KMT2ALMNAL3MBTL1
SCHEMBL16054078 0.78 HPGDS (0.45) USP30MEN1KMT2ALMNAL3MBTL1
SCHEMBL9892916 0.78 TP53 (0.60) USP30NPC1MEN1KMT2ALMNA
SCHEMBL16238715 0.77 L3MBTL1 (0.55) USP30NPC1MEN1KMT2ALMNA
SCHEMBL9892805 0.77 USP30 (0.48) USP30NPC1MEN1KMT2ALMNA
SCHEMBL13257796 0.77 L3MBTL1 (0.55) USP30NPC1MEN1KMT2ALMNA
SCHEMBL9892928 0.76 SMN1; SMN2 (0.56) USP30NPC1MEN1KMT2ALMNA
SCHEMBL4956602 0.75 TSHR (0.47) USP30MEN1KMT2ALMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8383615-B2 Azetidine 2-carboxamide derivatives which modulate the CB2 receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-02-26 US disclosed
US-20120142666-A1 Azetidine 2-Carboxamide Derivatives Which Modulate The CB2 Receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142666-A1 Azetidine 2-Carboxamide Derivatives Which Modulate The CB2 Receptor CNR2, CNR1, OPRL1 USP30 2593/4885NPC1 1689/4885MEN1 4667/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.