SCHEMBL9899749

SCHEMBL9899749

O=C(Nc1ccncc1-c1ccc(OS(=O)(=O)C(F)(F)F)cc1)OCCc1ccccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 3/20 0.42
IDH2 P48735 3/20 0.38
PTGS1 P23219 4/20 0.37
PTGS2 P35354 4/20 0.37
CHRM3 P20309 1/20 0.36
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
CHRNA7 P36544 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900135 0.84 BCL6 (0.39) CHRM3BCHEACHEMEN1KMT2A
SCHEMBL9899613 0.81 ROCK2 (0.43) SLC22A12IDH2CHRM3BCHEACHE
SCHEMBL9915915 0.80 LPAR1 (0.49) SLC22A12PTGS1PTGS2
SCHEMBL9899393 0.79 LPAR1 (0.40) CHRM3BCHEACHE
SCHEMBL9900012 0.77 CHRM3 (0.48) CHRM3
SCHEMBL9899562 0.75 BCHE (0.55) BCHEACHEMEN1KMT2ATRPV1
SCHEMBL15261910 0.69 LPAR1 (0.45) SLC22A12GSK3AGSK3B
SCHEMBL9915929 0.69 LPAR1 (0.45) SLC22A12GSK3AGSK3B
SCHEMBL7112369 0.67 CYP2A6 (0.50) PTGS1PTGS2
SCHEMBL27799850 0.63 HSD11B1 (0.43) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648714-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF Amira Pharmaceuticals, Inc. (US) 2013-10-16 EP disclosed
WO-2012078593-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF AMIRA PHARMACEUTICALS, INC. (US) 2012-06-14 WO disclosed