Bicarbonate

Bicarbonate

SCHEMBL9900307

COc1ccc(CC2CC2)cc1CNC(=O)c1ccc(Cl)cc1Cl.O=C(O)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.45
PPARG P37231 1/20 0.45
PPARD Q03181 1/20 0.45
PYGL P06737 2/20 0.45
LMNA P02545 2/20 0.44
HPGD P15428 1/20 0.44
RECQL P46063 2/20 0.43
POLB P06746 1/20 0.43
THRB P10828 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
DNMT3A Q9Y6K1 1/20 0.43
FLT1 P17948 1/20 0.43
FLT4 P35916 1/20 0.43
KDR P35968 1/20 0.43
TSHR P16473 1/20 0.43
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
SLC6A9 P48067 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5031740 0.81 PPARA (0.44) PPARAPPARGPPARDLMNAHPGD
SCHEMBL13433272 0.79 ALDH1A1 (0.52) PPARAPPARGPPARDLMNAHPGD
SCHEMBL6060870 0.78 PPARA (0.51) PPARAPPARGPPARD
SCHEMBL6493753 0.78 PPARA (0.58) PPARAPPARGPPARD
SCHEMBL6060873 0.78 PPARA (0.51) PPARAPPARGPPARD
SCHEMBL5034443 0.78 PPARA (0.42) PPARAPPARGPPARDPYGLLMNA
SCHEMBL3416041 0.77 LMNA (0.50) PPARAPPARGPPARDPYGLLMNA
SCHEMBL6495179 0.77 HPGD (0.67) PPARGLMNAHPGDRECQLPOLB
SCHEMBL14189965 0.77 PPARA (0.41) PPARAPPARGPPARDPYGLLMNA
SCHEMBL6504644 0.77 CYP1A2 (0.53) PYGLLMNAHPGDRECQLPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649045-B1 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2015-05-27 EP disclosed
EP-2649045-A2 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF Bayer Intellectual Property GmbH (DE) 2013-10-16 EP disclosed
WO-2012076466-A2 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-14 WO disclosed