SCHEMBL9901055

SCHEMBL9901055

O=C(O)N(c1cncc(Br)c1)C1CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38
SLC6A4 P31645 3/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TACR1 P25103 2/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CHRM3 P20309 1/20 0.34
ALOX15 P16050 1/20 0.34
HTT P42858 1/20 0.34
SMYD3 Q9H7B4 1/20 0.34
QPCT Q16769 1/20 0.34
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900770 0.81 NPC1 (0.40) SLC6A4SLC6A2SLC6A3TACR1NPC1
SCHEMBL2220667 0.75 HRH3 (0.38) POLBHCAR2HRH3CHRNB2CHRNA4
SCHEMBL8553350 0.72 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3ALDH1A1NPC1
SCHEMBL4441427 0.70 POLB (0.57) POLBHCAR2ALDH1A1NPC1RAB9A
SCHEMBL27369328 0.69 CHRM2 (0.47) SLC6A4SLC6A2SLC6A3TACR1CHRM3
SCHEMBL15367167 0.69 POLB (0.40) POLBHCAR2ALDH1A1NPC1RAB9A
SCHEMBL2349391 0.69 TACR1 (0.44) SLC6A4SLC6A2SLC6A3TACR1QPCT
SCHEMBL3507485 0.67 POLB (0.48) POLBHCAR2ALDH1A1NPC1RAB9A
SCHEMBL12504878 0.67 SLC6A4 (0.36) SLC6A4SLC6A2SLC6A3HRH3ALDH1A1
Hydrochloric Acid SCHEMBL4997661 0.67 SLC6A4 (0.41) SLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649065-A1 BICYCLIC COMPOUNDS AS PIM INHIBITORS Amgen Inc. (US) 2013-10-16 EP disclosed
WO-2012078777-A1 BICYCLIC COMPOUNDS AS PIM INHIBITORS AMGEN INC. (US) 2012-06-14 WO disclosed