SCHEMBL9901873

SCHEMBL9901873

CC1(C)CCC(NC(=NC#N)Nc2ccc(Cl)cc2)CC(C)(C)N1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.36
THRB P10828 1/20 0.34
ALDH1A1 P00352 4/20 0.33
KMT2A Q03164 3/20 0.33
CYP2C19 P33261 3/20 0.33
KDM4E B2RXH2 2/20 0.33
GAA P10253 2/20 0.33
CYP2C9 P11712 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.33
NPC1 O15118 1/20 0.33
EPHX1 P07099 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
EPHX2 P34913 3/20 0.32
CYP2D6 P10635 2/20 0.32
CYP1A2 P05177 1/20 0.32
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.31
CHRNA7 P36544 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9902217 0.92 KDM4E (0.38) USP30THRBALDH1A1KMT2ACYP2C19
SCHEMBL9902214 0.92 KDM4E (0.38) USP30THRBALDH1A1KMT2ACYP2C19
SCHEMBL16994489 0.89 P2RX7 (0.38) ALDH1A1KMT2ACYP2C19KDM4EGAA
SCHEMBL9901609 0.89 FPR2 (0.35) KMT2AKDM4EGAASMN1; SMN2LMNA
SCHEMBL9901606 0.89 FPR2 (0.35) KMT2AKDM4EGAASMN1; SMN2LMNA
SCHEMBL9902380 0.89 P2RX7 (0.37) THRBALDH1A1KMT2ACYP2C19KDM4E
SCHEMBL9902381 0.89 P2RX7 (0.37) THRBALDH1A1KMT2ACYP2C19KDM4E
SCHEMBL16994497 0.89 P2RX7 (0.37) THRBALDH1A1KMT2ACYP2C19KDM4E
SCHEMBL9902494 0.88 MEN1 (0.37) USP30ALDH1A1KMT2ACYP2C19CYP2C9
SCHEMBL9902498 0.88 MEN1 (0.37) USP30ALDH1A1KMT2ACYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649048-A1 MULTIFUNCTIONAL NITROXIDE DERIVATIVES AND USES THEREOF Radikal Therapeutics Inc. (US) 2013-10-16 EP disclosed
WO-2012077108-A1 MULTIFUNCTIONAL NITROXIDE DERIVATIVES AND USES THEREOF RADIKAL THERAPEUTICS INC. (US) 2012-06-14 WO disclosed