SCHEMBL9902192

SCHEMBL9902192

CC(NC(=O)OC(C)(C)C)C(C)C(=O)N1CC(C#N)C1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.42
CTSL P07711 3/20 0.42
CTSB P07858 2/20 0.42
CTSS P25774 9/20 0.39
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
JAK2 O60674 2/20 0.35
JAK1 P23458 2/20 0.35
JAK3 P52333 2/20 0.35
PREP P48147 1/20 0.35
TSHR P16473 1/20 0.34
TYK2 P29597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2378971 0.88 CTSK (0.44) CTSKCTSLCTSBCTSSCA1
SCHEMBL2491119 0.88 CTSK (0.44) CTSKCTSLCTSBCTSSCA1
SCHEMBL14755238 0.84 CTSK (0.41) CTSKCTSLCTSBCTSSJAK2
SCHEMBL14737063 0.83 JAK2 (0.45) CTSKCTSLCTSBCTSSCA1
SCHEMBL2377722 0.82 JAK1 (0.41) CTSKCTSLCTSBCTSSJAK2
SCHEMBL14738121 0.81 CTSK (0.53) CTSKCTSLCTSBCTSSTSHR
SCHEMBL14738854 0.79 CTSS (0.46) CTSKCTSLCTSBCTSSTSHR
SCHEMBL9279847 0.77 CTSK (0.44) CTSKCTSLCTSBCA1CA2
SCHEMBL14737016 0.75 CTSK (0.43) CTSKCTSLCTSBCTSSCA1
SCHEMBL9279883 0.74 TSHR (0.41) CTSKCTSLCTSBCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078802-A1 PREPARATION OF SUBSTITUTED-4,5-DIHYDROPYRROLO[4,3,2-de][2,6]NAPHTHYRIDIN-3(1H)-ONES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-06-14 WO disclosed