SCHEMBL9903397

SCHEMBL9903397

C[C@H]1CN(c2ccc3ncc(S(=O)(=O)c4cccc(C(F)(F)F)c4)cc3c2)CCN1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.41
PIK3CA P42336 1/20 0.40
AKR1B1 P15121 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
HTR7 P34969 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NR1H2 P55055 3/20 0.38
NR1H3 Q13133 3/20 0.38
GHSR Q92847 2/20 0.37
HSP90AA1 P07900 1/20 0.37
CXCR5 P32302 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9902830 0.88 HTR6 (0.48) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL9903819 0.86 HTR6 (0.45) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL9903836 0.83 HTR6 (0.42) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL5072337 0.83 HTR6 (0.56) HTR6PIK3CAAKR1B1KDM4EHTR1A
SCHEMBL5072339 0.83 HTR6 (0.56) HTR6PIK3CAAKR1B1KDM4EHTR1A
SCHEMBL17580665 0.83 PIK3CA (0.42) HTR6PIK3CAAKR1B1TRPV1KDM4E
SCHEMBL17580765 0.82 TRPV1 (0.39) HTR6PIK3CAAKR1B1TRPV1KDM4E
SCHEMBL9903063 0.82 HTR6 (0.43) HTR6PIK3CAALDH1A1HTR1ADRD2
SCHEMBL9903823 0.81 GRM5 (0.43) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL9903925 0.81 HTR6 (0.43) HTR6HTR1ADRD2HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1956004-B1 Quinoline derivatives and their use as 5-HT6 ligands GLAXO GROUP LTD (GB) 2012-06-13 EP claimed