SCHEMBL9903703

SCHEMBL9903703

Cc1cccc([C@@H]2CCNC(=O)O2)c1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.49
HTR2A P28223 1/20 0.39
HTR2B P41595 1/20 0.39
PKM P14618 1/20 0.38
PBRM1 Q86U86 1/20 0.36
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
MGLL Q99685 2/20 0.34
PARP1 P09874 1/20 0.34
PARP10 Q53GL7 1/20 0.34
PARP11 Q9NR21 1/20 0.34
GRM7 Q14831 1/20 0.34
CTSV O60911 2/20 0.33
CTSL P07711 2/20 0.33
CTSB P07858 2/20 0.33
CTSS P25774 2/20 0.33
CTSK P43235 2/20 0.33
CTSC P53634 2/20 0.33
CTSF Q9UBX1 2/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4306942 0.89 HTR2C (0.45) HTR2CHTR2AHTR2BPKMPBRM1
SCHEMBL5129808 0.89 HTR2C (0.45) HTR2CHTR2AHTR2BPKMPBRM1
SCHEMBL4310679 0.76 HTR2C (0.49) HTR2CHTR2AHTR2BPKMHTR6
SCHEMBL5125493 0.76 HTR2C (0.49) HTR2CHTR2AHTR2BPKMHTR6
SCHEMBL28957041 0.74 HTR2C (0.47) HTR2CPBRM1
SCHEMBL29698141 0.74 HTR2C (0.47) HTR2CPBRM1
SCHEMBL28957039 0.74 HTR2C (0.47) HTR2CPBRM1
SCHEMBL13394483 0.72 PKM (0.50) HTR2CPKMPBRM1DDB1CRBN
SCHEMBL14521456 0.71 MAOB (0.42)
SCHEMBL1705219 0.71 MAOB (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973546-B1 CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITORS MERCK SHARP & DOHME (US) 2012-06-13 EP disclosed